CATH Classification

Domain Context

CATH Clusters

Superfamily 3.40.630.30
Functional Family Diamine acetyltransferase 1

Enzyme Information

2.3.1.57
Diamine N-acetyltransferase.
based on mapping to UniProt P21673
Acetyl-CoA + an alkane-alpha,omega-diamine = CoA + an N-acetyldiamine.
-!- Acts on 1,3-diaminopropane, 1,5-diaminopentane, putrescine, spermidine (forming N(1)- and N(8)-acetylspermidine), spermine, N(1)- acetylspermidine and N(8)-acetylspermidine.

UniProtKB Entries (1)

P21673
SAT1_HUMAN
Homo sapiens
Diamine acetyltransferase 1

PDB Structure

PDB 2B4D
External Links
Method X-RAY DIFFRACTION
Organism Escherichia
Primary Citation
Structures of wild-type and mutant human spermidine/spermine N1-acetyltransferase, a potential therapeutic drug target
Bewley, M.C., Graziano, V., Jiang, J.S., Matz, E., Studier, F.W., Pegg, A.P., Coleman, C.S., Flanagan, J.M.
Proc.Natl.Acad.Sci.Usa