PDB Information

PDB6QMK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMus musculus
Primary Citation
Structure-Activity and Structure-Conformation Relationships of Aryl Propionic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1/Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1/NRF2) Protein-Protein Interaction.
Heightman, T.D., Callahan, J.F., Chiarparin, E., Coyle, J.E., Griffiths-Jones, C., Lakdawala, A.S., McMenamin, R., Mortenson, P.N., Norton, D., Peakman, T.M., Rich, S.J., Richardson, C., Rumsey, W.L., Sanchez, Y., Saxty, G., Willems, H.M.G., Wolfe 3rd, L., Woolford, A.J., Wu, Z., Yan, H., Kerns, J.K., Davies, T.G.
J.Med.Chem.
HeaderProtein Binding
Released2019-02-07
Resolution1.720
CATH Insert Date28 Apr, 2019

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Apr, 2019 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6qmkA00 29 Apr, 2019 2.120.10.80 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9Z2X8 KEAP1_MOUSE Mus musculus Kelch-like ECH-associated protein 1