PDB Information

PDB6HVV
MethodX-RAY DIFFRACTION
Host OrganismSaccharomyces cerevisiae S288C
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of Inhibitors Selective for Human Proteasome beta 2c or beta 2i Subunits.
Xin, B.T., Huber, E.M., de Bruin, G., Heinemeyer, W., Maurits, E., Espinal, C., Du, Y., Janssens, M., Weyburne, E.S., Kisselev, A.F., Florea, B.I., Driessen, C., van der Marel, G.A., Groll, M., Overkleeft, H.S.
J.Med.Chem.
HeaderHydrolase
Released2018-10-11
Resolution2.700
CATH Insert Date03 Feb, 2019

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
a 03 Feb, 2019 Chopped
A 03 Feb, 2019 Chopped
b 03 Feb, 2019 Chopped
B 03 Feb, 2019 Chopped
C 03 Feb, 2019 Chopped
D 03 Feb, 2019 Chopped
E 03 Feb, 2019 Chopped
F 03 Feb, 2019 Chopped
G 03 Feb, 2019 Chopped
H 03 Feb, 2019 Chopped
I 03 Feb, 2019 Chopped
J 03 Feb, 2019 Chopped
K 03 Feb, 2019 Chopped
L 03 Feb, 2019 Chopped
M 03 Feb, 2019 Chopped
N 03 Feb, 2019 Chopped
O 03 Feb, 2019 Chopped
P 03 Feb, 2019 Chopped
Q 03 Feb, 2019 Chopped
R 03 Feb, 2019 Chopped
S 03 Feb, 2019 Chopped
T 03 Feb, 2019 Chopped
U 03 Feb, 2019 Chopped
V 03 Feb, 2019 Chopped
W 03 Feb, 2019 Chopped
X 03 Feb, 2019 Chopped
Y 03 Feb, 2019 Chopped
Z 03 Feb, 2019 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
6hvva00 04 Feb, 2019 3.60.20.10 Assigned
6hvvA00 04 Feb, 2019 3.60.20.10 Assigned
6hvvb00 04 Feb, 2019 3.60.20.10 Assigned
6hvvB00 04 Feb, 2019 3.60.20.10 Assigned
6hvvC00 04 Feb, 2019 3.60.20.10 Assigned
6hvvD00 04 Feb, 2019 3.60.20.10 Assigned
6hvvE00 04 Feb, 2019 3.60.20.10 Assigned
6hvvF00 04 Feb, 2019 3.60.20.10 Assigned
6hvvG00 04 Feb, 2019 3.60.20.10 Assigned
6hvvH00 04 Feb, 2019 3.60.20.10 Assigned
6hvvI00 04 Feb, 2019 3.60.20.10 Assigned
6hvvJ00 04 Feb, 2019 3.60.20.10 Assigned
6hvvK00 04 Feb, 2019 3.60.20.10 Assigned
6hvvL00 04 Feb, 2019 3.60.20.10 Assigned
6hvvM00 04 Feb, 2019 3.60.20.10 Assigned
6hvvN00 04 Feb, 2019 3.60.20.10 Assigned
6hvvO00 04 Feb, 2019 3.60.20.10 Assigned
6hvvP00 04 Feb, 2019 3.60.20.10 Assigned
6hvvQ00 04 Feb, 2019 3.60.20.10 Assigned
6hvvR00 04 Feb, 2019 3.60.20.10 Assigned
6hvvS00 04 Feb, 2019 3.60.20.10 Assigned
6hvvT00 04 Feb, 2019 3.60.20.10 Assigned
6hvvU00 04 Feb, 2019 3.60.20.10 Assigned
6hvvV00 04 Feb, 2019 3.60.20.10 Assigned
6hvvW00 04 Feb, 2019 3.60.20.10 Assigned
6hvvX00 04 Feb, 2019 3.60.20.10 Assigned
6hvvY00 04 Feb, 2019 3.60.20.10 Assigned
6hvvZ00 04 Feb, 2019 3.60.20.10 Assigned

UniProtKB Entries (30)

Accession Gene ID Taxon Description
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P40306 PSB10_HUMAN Homo sapiens Proteasome subunit beta type-10
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P40306 PSB10_HUMAN Homo sapiens Proteasome subunit beta type-10
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5