PDB Information

PDB6HDQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Aiming to Miss a Moving Target: Bromo and Extra Terminal Domain (BET) Selectivity in Constrained ATAD2 Inhibitors.
Bamborough, P., Chung, C.W., Furze, R.C., Grandi, P., Michon, A.M., Watson, R.J., Mitchell, D.J., Barnett, H., Prinjha, R.K., Rau, C., Sheppard, R.J., Werner, T., Demont, E.H.
J. Med. Chem.
HeaderTranscription
Released2018-08-18
Resolution1.700
CATH Insert Date30 Sep, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 30 Sep, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6hdqA01 01 Oct, 2018 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4