PDB Information

PDB6CZV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine.
Kharenko, O.A., Patel, R.G., Brown, S.D., Calosing, C., White, A., Lakshminarasimhan, D., Suto, R.K., Duffy, B.C., Kitchen, D.B., McLure, K.G., Hansen, H.C., van der Horst, E.H., Young, P.R.
J. Med. Chem.
HeaderTranscription/Inhibitor
Released2018-04-09
Resolution1.880
CATH Insert Date30 Sep, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 30 Sep, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6czvA01 01 Oct, 2018 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4