PDB Information

PDB5TBI
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors.
Halby, L., Marechal, N., Pechalrieu, D., Cura, V., Franchini, D.M., Faux, C., Alby, F., Troffer-Charlier, N., Kudithipudi, S., Jeltsch, A., Aouadi, W., Decroly, E., Guillemot, J.C., Page, P., Ferroud, C., Bonnefond, L., Guianvarc'h, D., Cavarelli, J., Arimondo, P.B.
Philos.Trans.R.Soc.Lond.B Biol.Sci.
HeaderTransferase
Released2016-09-12
Resolution2.290
CATH Insert Date14 Nov, 2017

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped
C 14 Nov, 2017 Chopped
D 14 Nov, 2017 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5tbiA01 16 Dec, 2017 3.40.50.150 Assigned
5tbiA02 16 Dec, 2017 2.70.160.11 Assigned
5tbiB01 16 Dec, 2017 3.40.50.150 Assigned
5tbiB02 16 Dec, 2017 2.70.160.11 Assigned
5tbiC01 16 Dec, 2017 3.40.50.150 Assigned
5tbiC02 16 Dec, 2017 2.70.160.11 Assigned
5tbiD01 16 Dec, 2017 3.40.50.150 Assigned
5tbiD02 16 Dec, 2017 2.70.160.11 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1