PDB Information

PDB5M51
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-guided design of purine-based probes for selective Nek2 inhibition.
Coxon, C.R., Wong, C., Bayliss, R., Boxall, K., Carr, K.H., Fry, A.M., Hardcastle, I.R., Matheson, C.J., Newell, D.R., Sivaprakasam, M., Thomas, H., Turner, D., Yeoh, S., Wang, L.Z., Griffin, R.J., Golding, B.T., Cano, C.
Oncotarget
HeaderTransferase/Inhibitor
Released2016-10-20
Resolution1.900
CATH Insert Date20 Nov, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 21 Nov, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5m51A01 25 Nov, 2016 3.30.200.20 Assigned
5m51A02 25 Nov, 2016 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P51955 NEK2_HUMAN Homo sapiens Serine/threonine-protein kinase Nek2