PDB Information

PDB5LIA
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceMus musculus
Primary Citation
Discovery of potent inhibitors of the lysophospholipase autotaxin.
Shah, P., Cheasty, A., Foxton, C., Raynham, T., Farooq, M., Gutierrez, I.F., Lejeune, A., Pritchard, M., Turnbull, A., Pang, L., Owen, P., Boyd, S., Stowell, A., Jordan, A., Hamilton, N.M., Hitchin, J.R., Stockley, M., MacDonald, E., Quesada, M.J., Trivier, E., Skeete, J., Ovaa, H., Moolenaar, W.H., Ryder, H.
Bioorg. Med. Chem. Lett.
HeaderHydrolase
Released2016-07-14
Resolution1.920
CATH Insert Date20 Nov, 2016

PDB Images (6)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 21 Nov, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5liaA01 24 Nov, 2016 4.10.410.20 Assigned
5liaA02 24 Nov, 2016 4.10.410.20 Assigned
5liaA03 24 Nov, 2016 3.40.720.10 Assigned
5liaA04 24 Nov, 2016 3.40.570.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9R1E6 ENPP2_MOUSE Mus musculus Ectonucleotide pyrophosphatase/phosphodiesterase family member 2