PDB Information

PDB5KDH
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen.
Ayoub, A.M., Hawk, L.M.L., Herzig, R.J., Jiang, J., Wisniewski, A.J., Gee, C.T., Zhao, P., Zhu, J.Y., Berndt, N., Offei-Addo, N.K., Scott, T.G., Qi, J., Bradner, J.E., Ward, T.R., Schonbrunn, E., Georg, G.I., Pomerantz, W.C.K.
J. Med. Chem.
HeaderTranscription/Inhibitor
Released2016-06-08
Resolution1.500
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5kdhA01 10 Dec, 2017 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4