PDB Information

PDB5G5W
MethodX-RAY DIFFRACTION
Host OrganismTRICHOPLUSIA NI
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of Indazole Ethers as Novel, Potent, Non-Steroidal Glucocorticoid Receptor Modulators.
Hemmerling, M., Edman, K., Lepisto, M., Eriksson, A., Ivanova, S., Dahmen, J., Rehwinkel, H., Berger, M., Hendrickx, R., Dearman, M., Jensen, T.J., Wissler, L., Hansson, T.
Bioorg.Med.Chem.Lett.
HeaderHormone
Released2016-06-08
Resolution2.200
CATH Insert Date07 May, 2017

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5g5wA00 12 May, 2017 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2