PDB Information

PDB5G55
MethodX-RAY DIFFRACTION
Host OrganismUNIDENTIFIED
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of Novel 3-Quinoline Carboxamides as Potent, Selective and Orally Bioavailable Inhibitors of Ataxia Telangiectasia Mutated (Atm) Kinase.
Degorce, S.L., Barlaam, B., Cadogan, E., Dishington, A.P., Ducray, R., Glossop, S.C., Hassall, L.A., Lach, F., Lau, A., Mcguire, T.M., Nowak, T., Ouvry, G., Pike, K.G., Thomason, A.G.
J.Med.Chem.
HeaderTransferase
Released2016-05-20
Resolution2.450
CATH Insert Date14 Aug, 2016

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 15 Aug, 2016 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5g55A01 01 Sep, 2016 3.10.20.90 Assigned
5g55A02 01 Sep, 2016 2.60.40.150 Assigned
5g55A03 01 Sep, 2016 1.25.40.70 Assigned
5g55A04 01 Sep, 2016 3.30.1010.10 Assigned
5g55A05 01 Sep, 2016 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform