PDB Information

PDB5ENH
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain.
Cox, O.B., Krojer, T., Collins, P., Monteiro, O., Talon, R., Bradley, A., Fedorov, O., Amin, J., Marsden, B.D., Spencer, J., von Delft, F., Brennan, P.E.
Chem Sci
HeaderSignaling Protein
Released2015-11-09
Resolution1.950
CATH Insert Date08 May, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 May, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5enhA00 15 Jul, 2016 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q8WWQ0 PHIP_HUMAN Homo sapiens PH-interacting protein