PDB Information

PDB5DJP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Discovery of Novel Allosteric Non-Bisphosphonate Inhibitors of Farnesyl Pyrophosphate Synthase by Integrated Lead Finding.
Marzinzik, A.L., Amstutz, R., Bold, G., Bourgier, E., Cotesta, S., Glickman, J.F., Gotte, M., Henry, C., Lehmann, S., Hartwieg, J.C., Ofner, S., Pelle, X., Roddy, T.P., Rondeau, J.M., Stauffer, F., Stout, S.J., Widmer, A., Zimmermann, J., Zoller, T., Jahnke, W.
Chemmedchem
HeaderTransferase
Released2015-09-02
Resolution2.400
CATH Insert Date04 Oct, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
F 05 Oct, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5djpF00 01 Nov, 2015 1.10.600.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P14324 FPPS_HUMAN Homo sapiens Farnesyl pyrophosphate synthase