PDB Information

PDB5BWR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits.
Bertrand, S.M., Ancellin, N., Beaufils, B., Bingham, R.P., Borthwick, J.A., Boullay, A.B., Boursier, E., Carter, P.S., Chung, C.W., Churcher, I., Dodic, N., Fouchet, M.H., Fournier, C., Francis, P.L., Gummer, L.A., Herry, K., Hobbs, A., Hobbs, C.I., Homes, P., Jamieson, C., Nicodeme, E., Pickett, S.D., Reid, I.H., Simpson, G.L., Sloan, L.A., Smith, S.E., Somers, D.O., Spitzfaden, C., Suckling, C.J., Valko, K., Washio, Y., Young, R.J.
J.Med.Chem.
HeaderTransferase
Released2015-06-08
Resolution2.200
CATH Insert Date16 Aug, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped
B 17 Aug, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5bwrA01 24 Aug, 2015 3.30.470.10 Assigned
5bwrA02 24 Aug, 2015 3.20.10.10 Assigned
5bwrB01 24 Aug, 2015 3.30.470.10 Assigned
5bwrB02 24 Aug, 2015 3.20.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O15382 BCAT2_HUMAN Homo sapiens Branched-chain-amino-acid aminotransferase, mitochondrial
O15382 BCAT2_HUMAN Homo sapiens Branched-chain-amino-acid aminotransferase, mitochondrial