PDB Information

PDB5BRE
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceTrypanosoma cruzi (strain CL Brener)
Primary Citation
Structure-based approach to the identification of a novel group of selective glucosamine analogue inhibitors of Trypanosoma cruzi glucokinase.
D'Antonio, E.L., Deinema, M.S., Kearns, S.P., Frey, T.A., Tanghe, S., Perry, K., Roy, T.A., Gracz, H.S., Rodriguez, A., D'Antonio, J.
Mol.Biochem.Parasitol.
HeaderTransferase/Transferase Inhibitor
Released2015-05-30
Resolution2.500
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5breA01 27 Jul, 2015 3.30.420.40 Assigned
5breA02 27 Jul, 2015 3.40.367.20 Assigned
5breB01 27 Jul, 2015 3.30.420.40 Assigned
5breB02 27 Jul, 2015 3.40.367.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q4E4E1 Q4E4E1_TRYCC Trypanosoma cruzi strain CL Brener Glucokinase 1, putative
Q4E4E1 Q4E4E1_TRYCC Trypanosoma cruzi strain CL Brener Glucokinase 1, putative