PDB Information

PDB5AKU
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of Potent and Selective Nonplanar Tankyrase Inhibiting Nicotinamide Mimics.
Nkizinkiko, Y., Suneel Kumar, B.V.S., Jeankumar, V.U., Haikarainen, T., Koivunen, J., Madhuri, C., Yogeeswari, P., Venkannagari, H., Obaji, E., Pihlajaniemi, T., Sriram, D., Lehtio, L.
Bioorg.Med.Chem.
HeaderTransferase
Released2015-03-05
Resolution1.800
CATH Insert Date16 Aug, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped
B 17 Aug, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5akuA00 24 Aug, 2015 3.90.228.10 Assigned
5akuB00 24 Aug, 2015 3.90.228.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2