PDB Information

PDB4XX9
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Small-Molecule Allosteric Modulators of the Protein Kinase PDK1 from Structure-Based Docking.
Rettenmaier, T.J., Fan, H., Karpiak, J., Doak, A., Sali, A., Shoichet, B.K., Wells, J.A.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-01-30
Resolution1.400
CATH Insert Date08 Nov, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 Nov, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4xx9A01 12 Nov, 2015 3.30.200.20 Assigned
4xx9A02 12 Nov, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O15530 PDPK1_HUMAN Homo sapiens 3-phosphoinositide-dependent protein kinase 1