PDB Information

PDB4WRB
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design, synthesis, and protein crystallography of biaryltriazoles as potent tautomerase inhibitors of macrophage migration inhibitory factor.
Dziedzic, P., Cisneros, J.A., Robertson, M.J., Hare, A.A., Danford, N.E., Baxter, R.H., Jorgensen, W.L.
J.Am.Chem.Soc.
HeaderIsomerase/Isomerase Inhibitor
Released2014-10-23
Resolution1.810
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4wrbA00 22 Jul, 2015 3.30.429.10 Assigned
4wrbB00 20 Jul, 2015 3.30.429.10 Assigned
4wrbC00 22 Jul, 2015 3.30.429.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P14174 MIF_HUMAN Homo sapiens Macrophage migration inhibitory factor
P14174 MIF_HUMAN Homo sapiens Macrophage migration inhibitory factor
P14174 MIF_HUMAN Homo sapiens Macrophage migration inhibitory factor