PDB Information

PDB4WHZ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and Synthesis of Highly Potent and Isoform Selective JNK3 Inhibitors: SAR Studies on Aminopyrazole Derivatives.
Zheng, K., Iqbal, S., Hernandez, P., Park, H., LoGrasso, P.V., Feng, Y.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2014-09-24
Resolution1.790
CATH Insert Date07 Dec, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Dec, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4whzA01 28 Dec, 2014 3.30.200.20 Assigned
4whzA02 28 Dec, 2014 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P53779 MK10_HUMAN Homo sapiens Mitogen-activated protein kinase 10