PDB Information

PDB4QYF
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of the 1,7-diazacarbazole class of inhibitors of checkpoint kinase 1.
Gazzard, L., Appleton, B., Chapman, K., Chen, H., Clark, K., Drobnick, J., Goodacre, S., Halladay, J., Lyssikatos, J., Schmidt, S., Sideris, S., Wiesmann, C., Williams, K., Wu, P., Yen, I., Malek, S.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2014-07-24
Resolution2.150
CATH Insert Date28 Dec, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Dec, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4qyfA01 06 Jan, 2015 3.30.200.20 Assigned
4qyfA02 06 Jan, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14757 CHK1_HUMAN Homo sapiens Serine/threonine-protein kinase Chk1