PDB Information

PDB4QH6
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceTrypanosoma cruzi
Primary Citation
Molecular Design, Synthesis and Trypanocidal Activity of Dipeptidyl Nitriles as Cruzain Inhibitors.
Avelar, L.A., Camilo, C.D., de Albuquerque, S., Fernandes, W.B., Goncalez, C., Kenny, P.W., Leitao, A., McKerrow, J.H., Montanari, C.A., Orozco, E.V., Ribeiro, J.F., Rocha, J.R., Rosini, F., Saidel, M.E.
Plos Negl Trop Dis
HeaderHydrolase/Hydrolase Inhibitor
Released2014-05-27
Resolution3.130
CATH Insert Date16 Aug, 2015

PDB Images (11)

PDB Prints

PDB Chains (5)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped
B 17 Aug, 2015 Chopped
C 17 Aug, 2015 Chopped
D 17 Aug, 2015 Chopped
E 17 Aug, 2015 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
4qh6A00 20 Mar, 2016 3.90.70.10 Assigned
4qh6B00 20 Mar, 2016 3.90.70.10 Assigned
4qh6C00 20 Mar, 2016 3.90.70.10 Assigned
4qh6D00 20 Mar, 2016 3.90.70.10 Assigned
4qh6E00 20 Mar, 2016 3.90.70.10 Assigned

UniProtKB Entries (5)

Accession Gene ID Taxon Description
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain