PDB Information

PDB4PX6
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Syk inhibitors with high potency in presence of blood.
Thoma, G., Blanz, J., Buhlmayer, P., Druckes, P., Kittelmann, M., Smith, A.B., van Eis, M., Vangrevelinghe, E., Zerwes, H.G., Che, J.J., He, X., Jin, Y., Lee, C.C., Michellys, P.Y., Uno, T., Liu, H.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2014-03-21
Resolution1.600
CATH Insert Date27 Apr, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Apr, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4px6A01 03 May, 2014 3.30.200.20 Assigned
4px6A02 03 May, 2014 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P43405 KSYK_HUMAN Homo sapiens Tyrosine-protein kinase SYK