PDB Information

PDB4PCI
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of BRD4 bromodomain inhibitors by fragment-based high-throughput docking.
Zhao, H., Gartenmann, L., Dong, J., Spiliotopoulos, D., Caflisch, A.
Bioorg.Med.Chem.Lett.
HeaderTranscription/Transcription Inhibitor
Released2014-04-15
Resolution1.250
CATH Insert Date18 May, 2014

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 19 May, 2014 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4pciA01 21 May, 2014 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4