PDB Information

PDB4IR6
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B.
Chen, P., Chaikuad, A., Bamborough, P., Bantscheff, M., Bountra, C., Chung, C.W., Fedorov, O., Grandi, P., Jung, D., Lesniak, R., Lindon, M., Muller, S., Philpott, M., Prinjha, R., Rogers, C., Selenski, C., Tallant, C., Werner, T., Willson, T.M., Knapp, S., Drewry, D.H.
J.Med.Chem.
HeaderTranscription
Released2013-01-14
Resolution1.800
CATH Insert Date27 Jan, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Jan, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4ir6A00 01 Feb, 2013 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9UIF8 BAZ2B_HUMAN Homo sapiens Bromodomain adjacent to zinc finger domain protein 2B