PDB Information

PDB4IA9
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction.
Bolshan, Y., Getlik, M., Kuznetsova, E., Wasney, G.A., Hajian, T., Poda, G., Nguyen, K.T., Wu, H., Dombrovski, L., Dong, A., Senisterra, G., Schapira, M., Arrowsmith, C.H., Brown, P.J., Al-Awar, R., Vedadi, M., Smil, D.
ACS Med Chem Lett
HeaderTranscription
Released2012-12-06
Resolution1.660
CATH Insert Date30 Dec, 2012

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 31 Dec, 2012 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4ia9A00 17 Jul, 2013 2.130.10.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P61964 WDR5_HUMAN Homo sapiens WD repeat-containing protein 5