PDB 4i9u
PDB Information
PDB | 4I9U |
Method | X-RAY DIFFRACTION |
Host Organism | |
Gene Source | |
Primary Citation | Fragment growing and linking lead to novel nanomolar lactate dehydrogenase inhibitors.
J.Med.Chem.
|
Header | Oxidoreductase/Oxidoreductase Inhibitor |
Released | 2012-12-05 |
Resolution | 2.500 |
CATH Insert Date | 27 Jan, 2013 |
PDB Images (25)
PDB Prints
PDB Chains (8)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 28 Jan, 2013 | Chopped |
B | 28 Jan, 2013 | Chopped |
C | 28 Jan, 2013 | Chopped |
D | 28 Jan, 2013 | Chopped |
E | 28 Jan, 2013 | Chopped |
F | 28 Jan, 2013 | Chopped |
G | 28 Jan, 2013 | Chopped |
H | 28 Jan, 2013 | Chopped |
CATH Domains (16)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4i9uA01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uA02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
4i9uB01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uB02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
4i9uC01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uC02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
4i9uD01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uD02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
4i9uE01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uE02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
4i9uF01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uF02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
4i9uG01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uG02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
4i9uH01 | 02 Feb, 2013 | 3.40.50.720 | Assigned |
4i9uH02 | 02 Feb, 2013 | 3.90.110.10 | Assigned |
UniProtKB Entries (8)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |
P13491 | LDHA_RABIT | Oryctolagus cuniculus | L-lactate dehydrogenase A chain |