PDB Information

PDB4I9U
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Fragment growing and linking lead to novel nanomolar lactate dehydrogenase inhibitors.
Kohlmann, A., Zech, S.G., Li, F., Zhou, T., Squillace, R.M., Commodore, L., Greenfield, M.T., Lu, X., Miller, D.P., Huang, W.S., Qi, J., Thomas, R.M., Wang, Y., Zhang, S., Dodd, R., Liu, S., Xu, R., Xu, Y., Miret, J.J., Rivera, V., Clackson, T., Shakespeare, W.C., Zhu, X., Dalgarno, D.C.
J.Med.Chem.
HeaderOxidoreductase/Oxidoreductase Inhibitor
Released2012-12-05
Resolution2.500
CATH Insert Date27 Jan, 2013

PDB Images (25)

PDB Prints

PDB Chains (8)

Chain ID Date inserted into CATH CATH Status
A 28 Jan, 2013 Chopped
B 28 Jan, 2013 Chopped
C 28 Jan, 2013 Chopped
D 28 Jan, 2013 Chopped
E 28 Jan, 2013 Chopped
F 28 Jan, 2013 Chopped
G 28 Jan, 2013 Chopped
H 28 Jan, 2013 Chopped

CATH Domains (16)

Domain ID Date inserted into CATH Superfamily CATH Status
4i9uA01 02 Feb, 2013 3.40.50.720 Assigned
4i9uA02 02 Feb, 2013 3.90.110.10 Assigned
4i9uB01 02 Feb, 2013 3.40.50.720 Assigned
4i9uB02 02 Feb, 2013 3.90.110.10 Assigned
4i9uC01 02 Feb, 2013 3.40.50.720 Assigned
4i9uC02 02 Feb, 2013 3.90.110.10 Assigned
4i9uD01 02 Feb, 2013 3.40.50.720 Assigned
4i9uD02 02 Feb, 2013 3.90.110.10 Assigned
4i9uE01 02 Feb, 2013 3.40.50.720 Assigned
4i9uE02 02 Feb, 2013 3.90.110.10 Assigned
4i9uF01 02 Feb, 2013 3.40.50.720 Assigned
4i9uF02 02 Feb, 2013 3.90.110.10 Assigned
4i9uG01 02 Feb, 2013 3.40.50.720 Assigned
4i9uG02 02 Feb, 2013 3.90.110.10 Assigned
4i9uH01 02 Feb, 2013 3.40.50.720 Assigned
4i9uH02 02 Feb, 2013 3.90.110.10 Assigned

UniProtKB Entries (8)

Accession Gene ID Taxon Description
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain
P13491 LDHA_RABIT Oryctolagus cuniculus L-lactate dehydrogenase A chain