PDB Information

PDB4GTP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Development of Selective, Potent RabGGTase Inhibitors
Stigter, E.A., Guo, Z., Bon, R.S., Wu, Y.W., Choidas, A., Wolf, A., Menninger, S., Waldmann, H., Blankenfeldt, W., Goody, R.S.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2012-08-29
Resolution2.750
CATH Insert Date04 Nov, 2012

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped
B 05 Nov, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4gtpA00 10 Nov, 2012 1.25.40.120 Assigned
4gtpB00 08 Feb, 2013 1.50.10.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q04631 FNTA_RAT Rattus norvegicus Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha
Q02293 FNTB_RAT Rattus norvegicus Protein farnesyltransferase subunit beta