PDB Information

PDB4FHJ
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and optimization of potent and selective imidazopyridine and imidazopyridazine mTOR inhibitors.
Peterson, E.A., Boezio, A.A., Andrews, P.S., Boezio, C.M., Bush, T.L., Cheng, A.C., Choquette, D., Coats, J.R., Colletti, A.E., Copeland, K.W., Dupont, M., Graceffa, R., Grubinska, B., Kim, J.L., Lewis, R.T., Liu, J., Mullady, E.L., Potashman, M.H., Romero, K., Shaffer, P.L., Stanton, M.K., Stellwagen, J.C., Teffera, Y., Yi, S., Cai, T., La, D.S.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Inhibitor
Released2012-06-06
Resolution2.600
CATH Insert Date04 Nov, 2012

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
4fhjA01 10 Nov, 2012 3.10.20.90 Assigned
4fhjA02 10 Nov, 2012 2.60.40.150 Assigned
4fhjA03 10 Nov, 2012 1.25.40.70 Assigned
4fhjA04 10 Nov, 2012 3.30.1010.10 Assigned
4fhjA05 10 Nov, 2012 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform