PDB Information

PDB3ZVV
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHOMO SAPIENS
Primary Citation
Fragment based discovery of a novel and selective PI3 kinase inhibitor.
Hughes, S.J., Millan, D.S., Kilty, I.C., Lewthwaite, R.A., Mathias, J.P., O'Reilly, M.A., Pannifer, A., Phelan, A., Stuhmeier, F., Baldock, D.A., Brown, D.G.
Bioorg. Med. Chem. Lett.
HeaderTransferase
Released2011-07-27
Resolution2.500
CATH Insert Date02 Oct, 2011

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Nov, 2011 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
3zvvA01 04 Sep, 2013 3.10.20.90 Assigned
3zvvA02 04 Sep, 2013 2.60.40.150 Assigned
3zvvA03 04 Sep, 2013 1.25.40.70 Assigned
3zvvA04 04 Sep, 2013 3.30.1010.10 Assigned
3zvvA05 04 Sep, 2013 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform