PDB 3w5e
PDB Information
PDB | 3W5E |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Identification of the fused bicyclic 4-amino-2-phenylpyrimidine derivatives as novel and potent PDE4 inhibitors
Bioorg.Med.Chem.Lett.
|
Header | Hydrolase/Hydrolase Inhibitor |
Released | 2013-01-28 |
Resolution | 2.300 |
CATH Insert Date | 07 Jul, 2013 |
PDB Images (5)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 08 Jul, 2013 | Chopped |
B | 08 Jul, 2013 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
3w5eA00 | 09 Aug, 2013 | 1.10.1300.10 | Assigned |
3w5eB00 | 09 Aug, 2013 | 1.10.1300.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q07343 | PDE4B_HUMAN | Homo sapiens | cAMP-specific 3',5'-cyclic phosphodiesterase 4B |
Q07343 | PDE4B_HUMAN | Homo sapiens | cAMP-specific 3',5'-cyclic phosphodiesterase 4B |