PDB Information

PDB3U5J
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.
Filippakopoulos, P., Picaud, S., Fedorov, O., Keller, M., Wrobel, M., Morgenstern, O., Bracher, F., Knapp, S.
Bioorg.Med.Chem.
HeaderSignaling Protein/Inhibitor
Released2011-10-11
Resolution1.600
CATH Insert Date27 Nov, 2011

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Nov, 2011 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
3u5jA01 01 Dec, 2011 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4