PDB Information

PDB3QAR
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of triazine-benzimidazoles as selective inhibitors of mTOR.
Peterson, E.A., Andrews, P.S., Be, X., Boezio, A.A., Bush, T.L., Cheng, A.C., Coats, J.R., Colletti, A.E., Copeland, K.W., Dupont, M., Graceffa, R., Grubinska, B., Harmange, J.C., Kim, J.L., Mullady, E.L., Olivieri, P., Schenkel, L.B., Stanton, M.K., Teffera, Y., Whittington, D.A., Cai, T., La, D.S.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2011-01-11
Resolution2.650
CATH Insert Date03 Apr, 2011

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 04 Apr, 2011 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
3qarA01 04 Sep, 2013 3.10.20.90 Assigned
3qarA02 04 Sep, 2013 2.60.40.150 Assigned
3qarA03 04 Sep, 2013 1.25.40.70 Assigned
3qarA04 04 Sep, 2013 3.30.1010.10 Assigned
3qarA05 04 Sep, 2013 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform