PDB Information

PDB3PJ8
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Pyrazolo[4,3-d]pyrimidine Bioisostere of Roscovitine: Evaluation of a Novel Selective Inhibitor of Cyclin-Dependent Kinases with Antiproliferative Activity.
Jorda, R., McNae, I.W., Walkinshaw, M.D., Voller, J., Navratilova, J., Kuzma, M., Mistrik, M., Bartek, J., Strnad, M.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2010-11-09
Resolution1.960
CATH Insert Date10 Apr, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3pj8A01 11 Feb, 2013 3.30.200.20 Assigned
3pj8A02 11 Feb, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2