PDB Information

PDB3O57
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Pyrazolopyridines as potent PDE4B inhibitors: 5-heterocycle SAR.
Mitchell, C.J., Ballantine, S.P., Coe, D.M., Cook, C.M., Delves, C.J., Dowle, M.D., Edlin, C.D., Hamblin, J.N., Holman, S., Johnson, M.R., Jones, P.S., Keeling, S.E., Kranz, M., Lindvall, M., Lucas, F.S., Neu, M., Solanke, Y.E., Somers, D.O., Trivedi, N.A., Wiseman, J.O.
Bioorg.Med.Chem.Lett.
HeaderHydrolase/Hydrolase Inhibitor
Released2010-07-28
Resolution2.000
CATH Insert Date07 Aug, 2011

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Aug, 2011 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
3o57A00 25 Apr, 2013 1.10.1300.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q07343 PDE4B_HUMAN Homo sapiens cAMP-specific 3',5'-cyclic phosphodiesterase 4B