PDB Information

PDB3MG6
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S beta5-subunit.
Blackburn, C., Gigstad, K.M., Hales, P., Garcia, K., Jones, M., Bruzzese, F.J., Barrett, C., Liu, J.X., Soucy, T.A., Sappal, D.S., Bump, N., Olhava, E.J., Fleming, P., Dick, L.R., Tsu, C., Sintchak, M.D., Blank, J.L.
Biochem.J.
HeaderHydrolase
Released2010-04-05
Resolution2.600
CATH Insert Date22 May, 2011

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
1 23 May, 2011 Chopped
2 23 May, 2011 Chopped
A 23 May, 2011 Chopped
B 23 May, 2011 Chopped
C 23 May, 2011 Chopped
D 23 May, 2011 Chopped
E 23 May, 2011 Chopped
F 23 May, 2011 Chopped
G 23 May, 2011 Chopped
H 23 May, 2011 Chopped
I 23 May, 2011 Chopped
J 23 May, 2011 Chopped
K 23 May, 2011 Chopped
L 23 May, 2011 Chopped
M 23 May, 2011 Chopped
N 23 May, 2011 Chopped
O 23 May, 2011 Chopped
P 23 May, 2011 Chopped
Q 23 May, 2011 Chopped
R 23 May, 2011 Chopped
S 23 May, 2011 Chopped
T 23 May, 2011 Chopped
U 23 May, 2011 Chopped
V 23 May, 2011 Chopped
W 23 May, 2011 Chopped
X 23 May, 2011 Chopped
Y 23 May, 2011 Chopped
Z 23 May, 2011 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
3mg6100 26 May, 2011 3.60.20.10 Assigned
3mg6200 27 May, 2011 3.60.20.10 Assigned
3mg6A00 04 Feb, 2013 3.60.20.10 Assigned
3mg6B00 04 Feb, 2013 3.60.20.10 Assigned
3mg6C00 04 Feb, 2013 3.60.20.10 Assigned
3mg6D00 08 Feb, 2013 3.60.20.10 Assigned
3mg6E00 26 May, 2011 3.60.20.10 Assigned
3mg6F00 26 May, 2011 3.60.20.10 Assigned
3mg6G00 27 May, 2011 3.60.20.10 Assigned
3mg6H00 26 May, 2011 3.60.20.10 Assigned
3mg6I00 27 May, 2011 3.60.20.10 Assigned
3mg6J00 26 May, 2011 3.60.20.10 Assigned
3mg6K00 27 May, 2011 3.60.20.10 Assigned
3mg6L00 26 May, 2011 3.60.20.10 Assigned
3mg6M00 26 May, 2011 3.60.20.10 Assigned
3mg6N00 26 May, 2011 3.60.20.10 Assigned
3mg6O00 04 Feb, 2013 3.60.20.10 Assigned
3mg6P00 04 Feb, 2013 3.60.20.10 Assigned
3mg6Q00 04 Feb, 2013 3.60.20.10 Assigned
3mg6R00 08 Feb, 2013 3.60.20.10 Assigned
3mg6S00 27 May, 2011 3.60.20.10 Assigned
3mg6T00 26 May, 2011 3.60.20.10 Assigned
3mg6U00 26 May, 2011 3.60.20.10 Assigned
3mg6V00 27 May, 2011 3.60.20.10 Assigned
3mg6W00 27 May, 2011 3.60.20.10 Assigned
3mg6X00 27 May, 2011 3.60.20.10 Assigned
3mg6Y00 27 May, 2011 3.60.20.10 Assigned
3mg6Z00 27 May, 2011 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6