PDB Information

PDB3BIZ
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Synthesis and structure-activity relationships of soluble 8-substituted 4-(2-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-diones as inhibitors of the Wee1 and Chk1 checkpoint kinases.
Smaill, J.B., Lee, H.H., Palmer, B.D., Thompson, A.M., Squire, C.J., Baker, E.N., Booth, R.J., Kraker, A., Hook, K., Denny, W.A.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2007-12-02
Resolution2.200
CATH Insert Date27 Dec, 2007

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 27 Dec, 2007 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3bizA01 10 Sep, 2008 3.30.200.20 Assigned
3bizA02 10 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P30291 WEE1_HUMAN Homo sapiens Wee1-like protein kinase