PDB Information

PDB2XPA
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of Cell-Active Phenyl-Imidazole Pin1 Inhibitors by Structure-Guided Fragment Evolution.
Potter, A., Oldfield, V., Nunns, C., Fromont, C., Ray, S., Northfield, C.J., Bryant, C.J., Scrace, S.F., Robinson, D., Matossova, N., Baker, L., Dokurno, P., Surgenor, A.E., Davis, B., Richardson, C.M., Murray, J.B., Moore, J.D.
Bioorg.Med.Chem.Lett.
HeaderIsomerase
Released2010-08-25
Resolution1.900
CATH Insert Date23 Jan, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 24 Jan, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2xpaA01 17 Feb, 2011 2.20.70.10 Assigned
2xpaA02 17 Feb, 2011 3.10.50.40 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q13526 PIN1_HUMAN Homo sapiens Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1