PDB Information

PDB2RA0
MethodX-RAY DIFFRACTION
Host Organism
Gene SourceHomo sapiens
Primary Citation
7-fluoroindazoles as potent and selective inhibitors of factor xa.
Lee, Y.K., Parks, D.J., Lu, T., Thieu, T.V., Markotan, T., Pan, W., McComsey, D.F., Milkiewicz, K.L., Crysler, C.S., Ninan, N., Abad, M.C., Giardino, E.C., Maryanoff, B.E., Damiano, B.P., Player, M.R.
J.Med.Chem.
HeaderHydrolase
Released2007-09-14
Resolution2.300
CATH Insert Date21 Feb, 2008

PDB Images (6)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 21 Feb, 2008 Chopped
L 21 Feb, 2008 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
2ra0A01 23 Feb, 2008 2.40.10.10 Assigned
2ra0A02 23 Feb, 2008 2.40.10.10 Assigned
2ra0L00 22 Feb, 2008 2.10.25.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X